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Science/Engineering Conjugation Reactions In Drug Metabolism: An Integrated Approach by Gerard J. Mulder

Posted on 2010-03-16




Name:Science/Engineering Conjugation Reactions In Drug Metabolism: An Integrated Approach by Gerard J. Mulder
ASIN/ISBN:0850667380
Language:English
File size:3.01 Mb
Publisher: CRC Press
Publish Date: February 21, 1990
ISBN: 0850667380
Pages: 413
File Type: PDF
File Size: 3.01 MB
   Science/Engineering Conjugation Reactions In Drug Metabolism: An Integrated Approach by Gerard J. Mulder

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Conjugation Reactions In Drug Metabolism: An Integrated Approach by Gerard J. Mulder

This text investigates the molecular biology of conjugation, and the subsequent activity of the transfered genes "in vivo". Conjugation may be very important when considering biotransformations, as expression of transfered genes may allow organisms to metabolize certain substrates.

Contents

Preface v

Contributors vii

1. Introduction G.J.Mulder

2. Kinetics of conjugation reactions in eliminating organs K.S.Pang

3. Competition between conjugations for the same substrate G.J.Mulder

4. Glucuronidation G.J.Mulder, M.W.H.Coughtrie and B.Burchell

5. Sulfation G.J.Mulder and W.B.Jakoby

6. Acetylation W.W.Weber, G.N.Levy and D.W.Hein

7. O-Methylation D.R.Thakker and C.R.Creveling

8. N-Methyltransferases S.S.Ansher and W.B.Jakoby

9. S-Methylation J.L.Stevens and J.E.Bakke

10. Amino acid conjugation A.J.Hutt and J.Caldwell

11. Glutathione conjugation B.Ketterer and G.J.Mulder

12. Epoxide hydrolase T.M.Guenthner

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